PH17207A - New imidazo-rifamycin derivatives with antibacterial utility - Google Patents

New imidazo-rifamycin derivatives with antibacterial utility

Info

Publication number
PH17207A
PH17207A PH25656A PH25656A PH17207A PH 17207 A PH17207 A PH 17207A PH 25656 A PH25656 A PH 25656A PH 25656 A PH25656 A PH 25656A PH 17207 A PH17207 A PH 17207A
Authority
PH
Philippines
Prior art keywords
rifamycin derivatives
new imidazo
antibacterial utility
antibacterial
utility
Prior art date
Application number
PH25656A
Other languages
English (en)
Inventor
Egidio Marchi
Lauretta Montecchi
Original Assignee
Alfa Farmaceutici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfa Farmaceutici Spa filed Critical Alfa Farmaceutici Spa
Publication of PH17207A publication Critical patent/PH17207A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PH25656A 1980-05-22 1981-05-20 New imidazo-rifamycin derivatives with antibacterial utility PH17207A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT03429/80A IT1154655B (it) 1980-05-22 1980-05-22 Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica

Publications (1)

Publication Number Publication Date
PH17207A true PH17207A (en) 1984-06-19

Family

ID=11107198

Family Applications (2)

Application Number Title Priority Date Filing Date
PH25656A PH17207A (en) 1980-05-22 1981-05-20 New imidazo-rifamycin derivatives with antibacterial utility
PH26842A PH18704A (en) 1980-05-22 1982-02-09 Method of treatment using inidazo-rifamycin derivatives with antibacterial utility

Family Applications After (1)

Application Number Title Priority Date Filing Date
PH26842A PH18704A (en) 1980-05-22 1982-02-09 Method of treatment using inidazo-rifamycin derivatives with antibacterial utility

Country Status (25)

Country Link
US (1) US4341785A (en])
JP (1) JPS5711987A (en])
AR (1) AR226212A1 (en])
AT (1) AT373599B (en])
AU (1) AU537093B2 (en])
BE (1) BE888895A (en])
CA (1) CA1142518A (en])
CH (1) CH648037A5 (en])
DE (1) DE3120460A1 (en])
DK (1) DK157876C (en])
EG (1) EG14891A (en])
ES (1) ES502906A0 (en])
FI (1) FI69467C (en])
FR (1) FR2482967A1 (en])
GB (1) GB2079270B (en])
GR (1) GR75640B (en])
IE (1) IE51204B1 (en])
IT (1) IT1154655B (en])
LU (1) LU83376A1 (en])
NL (1) NL187022C (en])
NO (1) NO155622C (en])
PH (2) PH17207A (en])
PT (1) PT73064B (en])
SE (1) SE453089B (en])
ZA (1) ZA813430B (en])

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US20080262024A1 (en) * 2003-11-07 2008-10-23 Giuseppe Claudio Viscomi Rifaximin compositions and method of use
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US7256187B2 (en) * 2004-03-10 2007-08-14 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime derivatives effective against drug-resistant microbes
US7265107B2 (en) * 2004-03-10 2007-09-04 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes
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US8003118B2 (en) * 2005-03-02 2011-08-23 Kodsi Robert E Use of rifaximin for the prevention of aspiration pneumonia and/or sepsis
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KR101327635B1 (ko) 2005-08-11 2013-11-12 타간타 테라퓨틱스 인크. 포스폰산화 리파마이신, 및 그의 뼈 및 관절 감염의 저지및 치료 용도
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EP2054066B1 (en) 2006-08-02 2015-04-15 Salix Pharmaceuticals, Inc. Methods for treatment of radiation enteritis
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CA2663776C (en) * 2006-09-22 2016-01-26 Cipla Limited Rifaximin in an amorphous form
US20080161337A1 (en) * 2007-01-03 2008-07-03 Leonard Weinstock Use of Rifaximin for the Treatment of Chronic Prostatitis
US20080159987A1 (en) * 2007-01-03 2008-07-03 Leonard Weinstock Use of Rifaximin for the Treatment of Restless Legs Syndrome
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US11779571B2 (en) 2008-02-26 2023-10-10 Salix Pharmaceuticals, Inc. Methods for treating irritable bowel syndrome (IBS)
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EP2327407B1 (en) 2008-09-26 2014-07-09 ASKA Pharmaceutical Co., Ltd. Prophylactic and/or therapeutic agent for functional gastrointestinal disorders
US12285414B2 (en) 2008-10-02 2025-04-29 Salix Pharmaceuticals, Inc. Methods of treating hepatic encephalopathy
LT3628319T (lt) 2008-10-02 2024-03-25 Salix Pharmaceuticals, Inc. Hepatinės encefalopatijos gydymas rifaksiminu
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IT1397617B1 (it) * 2009-04-20 2013-01-18 Alfa Wassermann Spa Nuovi derivati della rifamicina
RU2540513C2 (ru) 2009-06-02 2015-02-10 Саликс Фармасьютикалз, Лтд. Способы лечения печеночной энцефалопатии
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KR20190000931A (ko) 2009-10-27 2019-01-03 루핀 리미티드 리팍시민의 고형 분산물
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US8952159B2 (en) 2009-12-28 2015-02-10 Silvio Massimo Lavagna Method for the production of amorphous rifaximin
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IT1398550B1 (it) 2010-03-05 2013-03-01 Alfa Wassermann Spa Formulazioni comprendenti rifaximina utili per ottenere un effetto prolungato nel tempo
JP6092629B2 (ja) 2010-03-10 2017-03-08 ルピン・リミテッドLupin Limited リファキシミン使用準備済懸濁液
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PH12013501643A1 (en) 2011-02-11 2019-10-11 Salix Pharmaceuticals Ltd Forms of rifaximin and uses thereof
EP2705042A1 (en) 2011-05-02 2014-03-12 Ranbaxy Laboratories Limited Rifaximin dimethylformamide solvate
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RU2496475C2 (ru) 2011-10-26 2013-10-27 Александр Васильевич Иващенко Фармацевтическая композиция и набор для лечения бактериальных инфекций
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JP2015509105A (ja) * 2012-01-25 2015-03-26 サリックス ファーマスーティカルズ,リミテッド リファキシミン誘導体及びその使用
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US9849090B2 (en) 2012-12-12 2017-12-26 Sun Pharmaceutical Industries Limited Pharmaceutical compositions of rifaximin
JP2016516988A (ja) 2013-03-15 2016-06-09 アルファ ワッセルマン ソシエタ ペル アチオニAlfa Wassermann S.P.A. 膣感染症を診断するための方法
US20160038468A1 (en) 2013-03-15 2016-02-11 Alfa Wassermann S.P.A. Rifaximin for use in the treating of vaginal infections
PL2983647T3 (pl) 2013-04-12 2021-01-25 Alfasigma S.P.A. Podawanie nlpz oraz związane z tym składniki, sposoby i układy
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CA2946101A1 (en) * 2014-04-19 2015-10-22 Granules India Limited An improved process for the preparation of rifamycin derivatives
JP6693946B2 (ja) 2014-05-04 2020-05-13 サリックス ファーマスーティカルズ,インコーポレーテッド Ibs微生物叢及びその使用
KR102362719B1 (ko) 2014-05-12 2022-02-14 알파시그마 에스.피.에이. 리팍시민의 신규한 용매화 결정 형태, 생산물, 조성물 및 이의 용도
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ES2868180T3 (es) 2017-06-26 2021-10-21 Biofer Spa Derivados de pirido-imidazo rifamicina como agentes antibacterianos
IT201700091912A1 (it) * 2017-08-08 2019-02-08 Biofer Spa Nuove pirido-imidazo rifamicine

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE273377C (en]) *
AT273377B (de) * 1967-03-01 1969-08-11 Lepetit Spa Verfahren zur Herstellung von neuen Rifamycinen
AT344898B (de) * 1975-06-13 1978-08-10 Archifar Ind Chim Trentino Verfahren zur herstellung neuer rifamycin-verbindungen
DK345977A (da) * 1976-09-30 1978-03-31 Archifar Ind Chim Trentino G rifamycinforbindelser og fremgangsmaade til deres fremstillin
CH629212A5 (it) * 1976-10-18 1982-04-15 Erba Farmitalia Procedimento per la preparazione di composti di rifamicina.
CH633014A5 (en) * 1978-06-09 1982-11-15 Erba Farmitalia Rifamycin compounds

Also Published As

Publication number Publication date
ES8203388A1 (es) 1982-04-01
ZA813430B (en) 1982-06-30
PH18704A (en) 1985-09-05
NO811731L (no) 1981-11-23
DE3120460A1 (de) 1982-03-11
IE811139L (en) 1981-11-22
US4341785A (en) 1982-07-27
GR75640B (en]) 1984-08-02
GB2079270A (en) 1982-01-20
NL187022B (nl) 1990-12-03
FR2482967A1 (fr) 1981-11-27
IT8003429A0 (it) 1980-05-22
FI811565L (fi) 1981-11-23
AU7065581A (en) 1981-11-26
NL187022C (nl) 1991-05-01
DK157876C (da) 1990-07-30
ES502906A0 (es) 1982-04-01
FI69467C (fi) 1986-02-10
IE51204B1 (en) 1986-10-29
LU83376A1 (fr) 1981-09-11
JPS5711987A (en) 1982-01-21
NO155622B (no) 1987-01-19
DK157876B (da) 1990-02-26
BE888895A (fr) 1981-09-16
JPS6123192B2 (en]) 1986-06-04
FI69467B (fi) 1985-10-31
EG14891A (en) 1985-12-31
CA1142518A (en) 1983-03-08
FR2482967B1 (en]) 1985-03-29
SE8103216L (sv) 1981-11-23
NO155622C (no) 1987-04-29
PT73064A (en) 1981-06-01
AU537093B2 (en) 1984-06-07
PT73064B (en) 1982-07-05
AT373599B (de) 1984-02-10
CH648037A5 (de) 1985-02-28
SE453089B (sv) 1988-01-11
GB2079270B (en) 1984-01-18
DE3120460C2 (en]) 1990-12-13
NL8102290A (nl) 1981-12-16
AR226212A1 (es) 1982-06-15
ATA222781A (de) 1983-06-15
DK224781A (da) 1981-11-23
IT1154655B (it) 1987-01-21

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